Results 1-20 of 20
Issue DateTitleAuthor(s)TypeМp-cat.
2025Pioneering first-in-class HDAC-ROCK inhibitors as potential multitarget anticancer agentsBeljkaš, Milan  ; Ružić, Dušan  ; Djurić, Ana  ; Vuletić, Ana  ; Nchugoua Tchiehe, Guilaine; Jallet, Corinne; Cadet-Daniel, Veronique; Arimondo, Paola B; Santibanez, Juan F.  ; Srdić-Rajić, Tatjana  ;
Nikolić, Katarina  ; Oljačić, Slavica  ; Petković, Miloš  ;
Article
22M22
2025Discovery of (3-Phenylcarbamoyl-3,4-dihydro-2H-pyrrol-2-yl)phosphonates as Imidazoline I2 Receptor Ligands with Anti-Alzheimer and Analgesic PropertiesBagán, Andrea; López-Ruiz, Alba; Abás, Sònia; Ruiz-Cantero, Carmen M.; Vasilopoulou, Foteini; Taboada-Jara, Teresa; Griñán-Ferré, Christian; Pallàs, Mercè; Muguruza, Carolina; Diez-Alarcia, , Rebeca;
Callado, Luis F.; Entrena, José M.; Cobos, Enrique J.; Pérez, Belén; Morales-García, José A.; Molins, Elies; De Jonghe, Steven; Daelemans, Dirk; Brea, José; Val, C.; Loza, M. Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Díaz, Caridad; Fernández-Godino, Rosario; Genilloud, Olga; Beljkaš, Milan  ; Oljačić, Slavica  ; Nikolić, Katarina  ; Escolano, Carmen;
Article
21a+M21a+
2025Određivanje strukture farmakofore, dizajn, sinteza i in vitro ispitivanje dualnih inhibitora histon deacetilaza (HDAC) i Rho-vezanih protein kinaza (ROCK)Beljkaš, Milan  Doctoral theses
70M70
2025Application of machine learning and molecular docking to the modelling and design of HDAC6/ROCK dual inhibitors with in vitro experimental validationBeljkaš, Milan  ; Zukić, Selma; Maran, Uko; Arimondo, Paola B; Petković, Miloš  ; Oljačić, Slavica  ; Nikolić, Katarina  Conference Paper
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2025P 01 Identification of Dual-Acting HDAC Inhibitors for Pancreatic Cancer Treatment through Drug Synergy Predictions and Molecular ModelingĐoković, Nemanja  ; Ilić, Aleksandra  ; Čebzan, Alen  ; Radović, Branko  ; Ružić, Dušan  ; Beljkaš, Milan  ; Đurić, Ana  ; Srdić-Rajić, Tatjana  ; Oljačić, Slavica  ; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2025Computer-Aided Drug Design of novel dual histone deacetylase inhibitorsIlić, Aleksandra  ; Beljkaš, Milan  ; Čebzan, Alen  ; Radović, Branko  ; Đoković, Nemanja  ; Nikolić, Katarina  ; Oljačić, Slavica  Conference Paper
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2025First Reported QSAR Models Of Dual HDAC6 And ROCK2 Inhibitors Employing Random Forest Regression AlgorithmZukić, Selma; Beljkaš, Milan  ; Maran, Uko; Petković, Miloš  ; Nikolić, Katarina  ; Oljačić, Slavica  Conference Paper
Mp. category will be shown later
2024Molecular modeling and design of new PI3K/HDAC dual inhibitorsBeljkaš, Milan  ; Kukić, E; Đoković, Nemanja  ; Oljačić, Slavica  Conference Paper
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2024Development of Novel ROCK Inhibitors via 3D-QSAR and Molecular Docking Studies: A Framework for Multi-Target Drug DesignBeljkaš, Milan  ; Petković, Miloš  ; Vuletić, Ana  ; Đurić, Ana  ; Santibanez, Juan F.  ; Srdić-Rajić, Tatjana  ; Nikolić, Katarina  ; Oljačić, Slavica  Article
21aM21a
2024Strengthening the epigenetic and signaling axis: Dual HDAC/ROCK inhibitors as a new therapeutic strategy in cancer treatmentBeljkaš, Milan  ; Petković, Miloš  ; Ružić, Dušan  ; Oljačić, Slavica  ; Nikolić, Katarina  ; Arimondo, Paola B; Srdić-Rajić, Tatjana  ; Vuletić, Ana  ; Jelić Mariokov Đurić, Ana  Conference Paper
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2024Discovery of dual-acting HDAC inhibitors for the treatment of pancreatic cancer by combining drug synergy and molecular modelingĐoković, Nemanja  ; Ilić, Aleksandra  ; Čebzan, Alen  ; Radović, Branko  ; Ružić, Dušan  ; Beljkaš, Milan  ; Đurić, Ana  ; Srdić-Rajić, Tatjana  ; Oljačić, Slavica  ; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2023Virtual docking and design of novel Histone deacetylase and Rho- associated protein kinases dual inhibitors (HDAC/ROCKs)Beljkaš, Milan  ; Petković, Miloš  ; Nikolić, Katarina  ; Oljačić, Slavica  Conference Paper
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2023Targeting Histone Deacetylases 6 in Dual-Target Therapy of CancerBeljkas, Milan  ; Ilić, Aleksandra  ; Cebzan, Alen  ; Radović, Branko  ; Đoković, Nemanja  ; Ružić, Dušan  ; Nikolić, Katarina  ; Oljačić, Slavica  Article
21aM21a
2023Virtual Docking, design and in silico ADMET profiling of novel Rho- associated protein kinases-1 (ROCK1) inhibitorsBeljkaš, Milan  ; Rebić, Jelena; Radan, Milica  ; Đikić, Teodora ; Oljačić, Slavica  ; Nikolić, Katarina  Conference Paper
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20233D-Quantitative Structure-Activity Relationship and design of novel Rho- associated protein kinases-1 (ROCK1) inhibitorsBeljkaš, Milan  ; Rebić, Jelena; Radan, Milica  ; Đikić, Teodora ; Oljačić, Slavica  ; Nikolić, Katarina  Conference Paper
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2023Preclinical Evaluation of an Imidazole-Linked Heterocycle for Alzheimer’s DiseaseBagán, Andrea; Rodriguez-Arévalo, Sergio; Taboada-Jara, Teresa; Griñán-Ferré, Christian; Pallàs, Mercè; Brocos-Mosquera, Iria; Callado, Luis F.; Morales-García, José A.; Pérez, Belén; Diaz, Caridad;
Fernández-Godino, Rosario; Genilloud, Olga; Beljkaš, Milan  ; Oljačić, Slavica  ; Nikolić, Katarina  ; Escolano, Carmen;
Article
21aM21a
20233D-Quantitative Structure-Activity Relationship approach in the design of novel Rho-associated protein kinases(ROCK) inhibitorsBeljkaš, Milan  ; Oljačić, Slavica  ; Petković, Miloš  ; Nikolić, Katarina  Conference Paper
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2022Discovery of 1-Benzhydryl-Piperazine-Based HDAC Inhibitors with Anti-Breast Cancer Activity: Synthesis, Molecular Modeling, In Vitro and In Vivo Biological EvaluationRužić, Dušan  ; Ellinger, Bernhard; Đoković, Nemanja  ; Santibanez, Juan  ; Gul, Sheraz; Beljkaš, Milan  ; Đurić, Ana  ; Ganesan, Arasu; Pavić, Aleksandar  ; Srdić-Rajić, Tatjana  ;
Petković, Miloš  ; Nikolić, Katarina  ;
Article
21aM21a
2022Anticancer evaluation of the selected tetrahydropyrimidines: 3D-QSAR, cytotoxic activities, mechanism of action, DNA, and BSA interactionsMilović Emilija  ; Petronijević Jelena  ; Joksimović Nenad  ; Beljkaš M.  ; Ružić D.  ; Nikoletić Katarina  ; Vraneš Milan  ; Tot Aleksandar S. ; Đorđić Crnogorac Marija  ; Stanojković Tatjana P.  ;
Janković Nenad  ;
Article
22M22
2019Is there a borderline between cytotoxic and antimetastatic effects of selective Histone deacetylase 6 inhibitors in solid malignancies?Nikolić, Katarina M.  ; Ružić, Dušan B.  ; Milan Beljkas  ; Petković, Miloš R.  ; Sheraz Gul; Juan F. Santibanez; Srdić-Rajić, Tatjana V.  Conference Paper
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