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Browsing by Author Burnett, James C.

Showing results 1 to 10 of 10
Issue DateTitleAuthor(s)TypeМ-cat.
20134-Amino-7-chloroquinolines: Probing Ligand Efficiency Provides Botulinum Neurotoxin Serotype A Light Chain Inhibitors with Significant Antiprotozoal ActivityOpsenica, Igor  ; Tot, Mikloš; Gomba, Laura; Nuss, Jonathan E.; Sciotti, Richard J.; Bavari, Sina; Burnett, James C.; Šolaja, Bogdan A. Article
21aM21a
2011A Chemotype That Inhibits Three Unrelated Pathogenic Targets: The Botulinum Neurotoxin Serotype A Light Chain, P. falciparum Malaria, and the Ebola Filovirus (✓)Opsenica, Igor  ; Burnett, James C.; Gussio, Rick; Opsenica, Dejan M.  ; Todorović, Nina  ; Lanteri, Charlotte A.; Sciotti, Richard J.; Gettayacamin, Montip; Basilico, Nicoletta; Taramelli, Donatella;
Nuss, Jonathan E.; Wanner, Laura; Panchal, Rekha G.; Šolaja, Bogdan A. ; Bavari, Sina;
Article
21aM21a
2012A Limited Structural Modification Results in a Significantly More Efficacious Diazachrysene-Based Filovirus Inhibitor (✓)Selaković, Života  ; Opsenica, Dejan M.  ; Eaton, Brett; Retterer, Cary; Bavari, Sina; Burnett, James C.; Šolaja, Bogdan A. ; Panchal, Rekha G.Article
22M22
2007A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype a metalloprotease (✓)Burnett, James C.; Opsenica, Dejan M.  ; Sriraghavan, Kamaraj; Panchal, Rekha G.; Ruthel, Gordon; Hermone, Ann R.; Nguyen, Tam L.; Kenny, Tara A.; Lane, Douglas J.; McGrath, Connor F.;
Schmidt, James J.; Vennerstrom, Jonathan L.; Gussio, Rick; Šolaja, Bogdan A. ; Bavari, Sina;
Article
21aM21a
2013Correlation between structure, retention, property, and activity of biologically relevant 1,7-bis(aminoalkyl)diazachrysene derivatives (✓)Šegan, Sandra B.  ; Trifković, Jelena  ; Verbić, Tatjana  ; Opsenica, Dejan M.  ; Zlatović, Mario  ; Burnett, James C.; Šolaja, Bogdan A. ; Milojković-Opsenica, Dušanka  Article
21M21
2013New 9-aminoacridine derivatives as inhibitors of botulinum neurotoxins and P. falciparum malaria (✓)Tot, Miklos; Opsenica, Dejan  ; Mitrić, Milena; Burnett, James C.; Gomba, Laura; Bavari, Sina; Šolaja, Bogdan Article
23M23
2008Novel 4-aminoquinolines active against chloroquine-resistant and sensitive P. falciparum strains that also inhibit botulinum serotype A (✓)Šolaja, Bogdan A. ; Opsenica, Dejan M.  ; Smith, Kirsten S.; Milhous, Wilbur K.; Terzić-Jovanović, Nataša  ; Opsenica, Igor  ; Burnett, James C.; Nuss, Jon; Gussio, Rick; Bavari, SinaArticle
21aM21a
2014Second Generation Steroidal 4-Aminoquinolines Are Potent, Dual-Target Inhibitors of the Botulinum Neurotoxin Serotype A Metalloprotease and P. falciparum Malaria (✓)Videnović, Milica  ; Opsenica, Dejan M.  ; Burnett, James C.; Gomba, Laura; Nuss, Jonathan E.; Selaković, Života  ; Konstantinović, Jelena M.  ; Krstić-Ristivojević, Maja  ; Šegan, Sandra B.  ; Zlatović, Mario  ;
Sciotti, Richard J.; Bavari, Sina; Šolaja, Bogdan A. ;
Article
21aM21a
2012The synthesis of 2,5-bis(4-amidinophenyl)thiophene derivatives providing submicromolar-range inhibition of the botulinum neurotoxin serotype A metalloprotease (✓)Opsenica, Igor  ; Filipović, Vuk  ; Nuss, Jon E.; Gomba, Laura M.; Opsenica, Dejan  ; Burnett, James C.; Gussio, Rick; Šolaja, Bogdan ; Bavari, SinaArticle
21M21
2008Three-Dimensional Database Mining Identifies a Unique Chemotype that Unites Structurally Diverse Botulinum Neurotoxin Serotype A Inhibitors in a Three-Zone PharmacophoreHermone, Ann R.; Burnett, James C.; Nuss, Jonathan E.; Tressler, Lyal E.; Nguyen, Tam L.; Šolaja, Bogdan A. ; Vennerstrom, Jonathan L.; Schmidt, James J.; Wipf, Peter; Bavari, Sina;
Gussio, Rick;
Article
21M21