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Browsing by Author Gussio, Rick
Showing results 1 to 5 of 5
Issue Date | Title | Author(s) | Type | М-cat. |
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2011 | A Chemotype That Inhibits Three Unrelated Pathogenic Targets: The Botulinum Neurotoxin Serotype A Light Chain, P. falciparum Malaria, and the Ebola Filovirus (✓) | Opsenica, Igor ; Burnett, James C.; Gussio, Rick; Opsenica, Dejan M. ; Todorović, Nina ; Lanteri, Charlotte A.; Sciotti, Richard J.; Gettayacamin, Montip; Basilico, Nicoletta; Taramelli, Donatella; | Article | 21aM21a |
2007 | A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype a metalloprotease (✓) | Burnett, James C.; Opsenica, Dejan M. ; Sriraghavan, Kamaraj; Panchal, Rekha G.; Ruthel, Gordon; Hermone, Ann R.; Nguyen, Tam L.; Kenny, Tara A.; Lane, Douglas J.; McGrath, Connor F.; | Article | 21aM21a |
2008 | Novel 4-aminoquinolines active against chloroquine-resistant and sensitive P. falciparum strains that also inhibit botulinum serotype A (✓) | Šolaja, Bogdan A. ; Opsenica, Dejan M. ; Smith, Kirsten S.; Milhous, Wilbur K.; Terzić-Jovanović, Nataša ; Opsenica, Igor ; Burnett, James C.; Nuss, Jon; Gussio, Rick; Bavari, Sina | Article | 21aM21a |
2012 | The synthesis of 2,5-bis(4-amidinophenyl)thiophene derivatives providing submicromolar-range inhibition of the botulinum neurotoxin serotype A metalloprotease (✓) | Opsenica, Igor ; Filipović, Vuk ; Nuss, Jon E.; Gomba, Laura M.; Opsenica, Dejan ; Burnett, James C.; Gussio, Rick; Šolaja, Bogdan ; Bavari, Sina | Article | 21M21 |
2008 | Three-Dimensional Database Mining Identifies a Unique Chemotype that Unites Structurally Diverse Botulinum Neurotoxin Serotype A Inhibitors in a Three-Zone Pharmacophore | Hermone, Ann R.; Burnett, James C.; Nuss, Jonathan E.; Tressler, Lyal E.; Nguyen, Tam L.; Šolaja, Bogdan A. ; Vennerstrom, Jonathan L.; Schmidt, James J.; Wipf, Peter; Bavari, Sina;
Gussio, Rick;
| Article | 21M21 |