Researchers



Results 21-40 of 92
Issue DateTitleAuthor(s)TypeМp-cat.
2023Computer-aided drug design of MAPK inhibitors by combined 3D-QSAR analysis and molecular dockingČebzan, Alen  ; Ružić, Dušan  ; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2022Design of Dual COX-2 and 5-LOX Inhibitors with Iron-Chelating Properties Using Structure-Based and Ligand-Based MethodsBošković, Jelena  ; Ružić, Dušan  ; Čudina, Olivera  ; Nikolic, Katarina  ; Dobričić, Vladimir  Article
23M23
2022Bistable Photoswitch Allows in Vivo Control of HematopoiesisAlbert, Lea; Nagpal, Jatin; Steinchen, Wieland; Zhang, Lei; Werel, Laura; Đoković, Nemanja  ; Ružić, Dušan  ; Hoffarth, Malte; Xu, Jing; Kaspareit, Johanna;
Abendroth, Frank; Royant, Antoine; Bange, Gert; Nikolić, Katarina  ; Ryu, Soojin; Dou, Yali; Essen, Lars-Oliver; Vázquez, Olalla;
Article
21a+M21a+
2022Dual LSD1 and HDAC6 Inhibition Induces Doxorubicin Sensitivity in Acute Myeloid Leukemia CellsBulut, Ipek; Lee, Adam; Cevatemre, Buse; Ružić, Dušan  ; Belle, Roman; Kawamura, Akane; Gul, Sheraz; Nikolić, Katarina  ; Ganesan, A.; Acilan, CeydaArticle
21M21
2022Novel protocol for enhanced sampling of binding pocket dynamics and its integration into the sirtuin 2 inhibitors virtual screening campaignĐoković, Nemanja  ; Ružić, Dušan  ; Rahnasto‐Rilla, Minna; Srdić-Rajić, Tatjana  ; Lahtela‐Kakkonen, Maija; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2022Epigenetic drug discovery: fragment-based drug design of novel 1-benzhydryl-piperazine derivatives as selective histone deacetylase 6 inhibitorsRužić, Dušan  ; Đoković, Nemanja  ; Srdić-Rajić, Tatjana  ; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2022Quinazoline-based analog of adenine as an antidote against MLL-rearranged leukemia cells: synthesis, inhibition assays and docking studiesBon, Corentin; Barbachowska, Magdalena; Đoković, Nemanja  ; Ružić, Dušan  ; Si, Yang; Soresinetti, Laura; Jallet, Corinne; Tafit, Ambre; Halby, Ludovic; Nikolić, Katarina  ;
Arimondo, Paola B;
Article
21M21
2022Design of novel dual COX 2 and 5 LOX inhibitors using quantitative structure activity relationships analysisBošković, Jelena  ; Dobričić, Vladimir  ; Ružić, Dušan  ; Nikolić, Katarina  ; Čudina, Olivera  Conference Paper
Mp. category will be shown later
2022Anticancer evaluation of the selected tetrahydropyrimidines: 3D-QSAR, cytotoxic activities, mechanism of action, DNA, and BSA interactionsMilović Emilija  ; Petronijević Jelena  ; Joksimović Nenad  ; Beljkaš M.  ; Ružić D.  ; Nikoletić Katarina  ; Vraneš Milan  ; Tot Aleksandar S. ; Đorđić Crnogorac Marija  ; Stanojković Tatjana P.  ;
Janković Nenad  ;
Article
22M22
2022Targeting Histone Deacetylases: Opportunities for Cancer Treatment and ChemopreventionRužić, Dušan  ; Đoković, Nemanja  ; Srdić-Rajić, Tatjana  ; Echeverria, Cesar; Nikolić, Katarina  ; Santibanez, Juan  Article
21aM21a
2022Racionalni dizajn, sinteza i in vitro ispitivanja selektivnih inhibitora histon deacetilaze 6Ružić, Dušan  Doctoral theses
70M70
2022Identification of novel 1-benzhydryl-piperazine derivatives as Histone Deacetylase inhibitors using Fragment-based drug design strategyRužić, Dušan  ; Ellinger, Bernhard; Đoković, Nemanja  ; Santibanez, Juan  ; Ganesan, A.; Pavić, Aleksandar; Srdić Rajić, Tatjana  ; Petković, Miloš  ; Nikolić, Katarina  Other
Mp. category will be shown later
2022Computer-aided drug design and evaluation of selective inhibitors against cytoplasmic histone deacetylasesRužić, Dušan  ; Đoković, Nemanja  ; Petković, Miloš  ; Gul, Sheraz; Lahtela‐Kakkonen, Maija; Ganesan, A.; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2022Discovery of 1-Benzhydryl-Piperazine-Based HDAC Inhibitors with Anti-Breast Cancer Activity: Synthesis, Molecular Modeling, In Vitro and In Vivo Biological EvaluationRužić, Dušan  ; Ellinger, Bernhard; Đoković, Nemanja  ; Santibanez, Juan  ; Gul, Sheraz; Beljkaš, Milan  ; Đurić, Ana  ; Ganesan, Arasu; Pavić, Aleksandar  ; Srdić-Rajić, Tatjana  ;
Petković, Miloš  ; Nikolić, Katarina  ;
Article
21aM21a
2022Rational design and in vitro evaluation of selective inhibitors of cytoplasmic histone deacetylases SIRT2 and HDAC6Ružić, Dušan  ; Đoković, Nemanja  ; Petković, Miloš  ; Gul, Sheraz; Lahtela‐Kakkonen, Maija; Ganesan, A.; Srdić-Rajić, Tatjana  ; Nikolić, Katarina  Conference Paper
Mp. category will be shown later
2022Expanding the Accessible Chemical Space of SIRT2 Inhibitors through Exploration of Binding Pocket DynamicsĐoković, Nemanja  ; Ružić, Dušan  ; Rahnasto-Rilla, Mina; Srdić-Rajić, Tatjana  ; Lahtela-Kakkonen, Maija; Nikolić, Katarina  Article
21aM21a
2021Synthesis and biological activity of a cytostatic inhibitor of MLLr leukemia targeting the DOT1L proteinBon, Corentin; Si, Yang; Pernak, Melanie; Barbachowska, Magdalena; Levi-Acobas, Eva; Cadet Daniel, Veronique; Jallet, Corinne; Ružić, Dušan  ; Đoković, Nemanja  ; Đikić, Teodora ;
Nikolić, Katarina  ; Halby, Ludovic; Arimondo, Paola B.;
Article
21M21
2021Epigenetic drug discovery: Successful examples of Computer-Aided Drug Designing of Histone Deacetylase (HDAC6 and SIRT2) and Histone Methyltransferase (DOT1L) inhibitorsRuzic, Dušan  ; Đoković, Nemanja B.  ; Bon C.; Petkovic, M.  ; Ellinger B.; Gul, S.; Santibanez F. J.; Lahtela-Kakkonen, M.; Halby L.; Ganesan, A.;
Srdic-Rajic T.  ; Arimondo P.; Nikolić, Katarina M.  ;
Conference Paper
Mp. category will be shown later
2021Fragment-Based Drug Design of Selective HDAC6 InhibitorsRužić, PhD, Dušan  Book parts
Mp. category will be shown later
2021An Integrative in silico Drug Repurposing Approach for Identification of Potential Inhibitors of SARS-CoV-2 Main ProteaseĐoković, Nemanja  ; Ružić, Dušan  ; Đikić, Teodora ; Cvijić, Sandra  ; Ignjatović, Jelisaveta ; Ibrić, Svetlana  ; Baralić, Katarina  ; Buha-Đorđević, Aleksandra  ; Ćurčić, Marijana  ; Đukić-Ćosić, Danijela  ;
Nikolić, Katarina  ;
Article
21M21