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Резултати

Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model   [2020]

Horatscheck, Andre; Andrijevic, Ana  ; Nchinda, Aloysius T.; Le Manach, Claire; Paquet, Tanya; Khonde, Lutete Peguy; Dam, Jean; Pawar, Kailash; Taylor, Dale; Lawrence, Nina;
Brunschwig, Christel; Gibhard, Liezl; Njoroge, Mathew; Reader, Janette; van der Watt, Mariette; Wicht, Kathryn; de Sousa, Ana Carolina C.; Okombo, John; Maepa, Keletso; Egan, Timothy J.; Birkholtz, Lyn-Marie; Basarab, Gregory S.; Wittlin, Sergio; Fish, Paul, V; Street, Leslie J.; Duffy, James; Chibale, Kelly;

Tetraoxane antimalarials and their reaction with Fe(II) (✓)   [2006]

Opsenica, Igor  ; Terzić-Jovanović, Nataša  ; Opsenica, Dejan M.  ; Angelovski, Goran ; Lehnig, Manfred; Eilbracht, Peter; Tinant, Bernard; Juranić, Zorica D.  ; Smith, Kirsten S.; Yang, Young S.;
Diaz, Damaris S.; Smith, Philip L.; Milhous, Wilbur K.; Dokovic, Dejan; Šolaja, Bogdan A. ;

Erratum: Bicyclic α-Iminophosphonates as High Affinity Imidazoline I2Receptor Ligands for Alzheimer's Disease (Journal of Medicinal Chemistry (2020) 63:7 (3610−3633) DOI: 10.1021/acs.jmedchem.9b02080)   [2020]

Abás, Sònia; Rodríguez-Arévalo, Sergio; Bagán, Andrea; Griñán-Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins, Elies; Luque, F. Javier;
Pérez-Lozano, Pilar; De Jonghe, Steven; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, M. Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica  ; Đikić, Teodora  ; Nikolić, Katarina  ; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmen;

Deoxycholic acid-derived tetraoxane antimalarials and antiproliferatives (✓)   [2007]

Terzić-Jovanović, Nataša  ; Opsenica, Dejan M.  ; Milić, Dragana  ; Tinant, Bernard; Smith, Kirsten S.; Milhous, Wilbur K.; Šolaja, Bogdan A. 

New Steroidal 4-Aminoquinolines Antagonize Botulinum Neurotoxin Serotype A in Mouse Embryonic Stem Cell Derived Motor Neurons in Postintoxication Model   [2018]

Konstantinović, Jelena M.  ; Kiris, Erkan; Kota, Krishna P.; Kugelman-Tonos, Johanny; Videnović, Milica  ; Cazares, Lisa H.; Terzić-Jovanović, Nataša  ; Verbić, Tatjana  ; Anđelković, Boban D.  ; Duplantier, Allen J.;
Bavari, Sina; Šolaja, Bogdan ;

2-[(Carboxymethyl)sulfanyl]-4-oxo-4-arylbutanoic acids selectively suppressed proliferation of neoplastic human HeLa cells. A SAR/QSAR study (✓)   [2005]

Drakulić, Branko J.; Juranić, Zorica D.  ; Stanojković, Tatjana P.  ; Ivan Juranic  

New Water-Soluble Copper(II) Complexes with Morpholine–Thiosemicarbazone Hybrids: Insights into the Anticancer and Antibacterial Mode of Action   [2018]

Ohui, Kateryna; Afanasenko, Eleonora; Bacher, Felix; Ting, Rachel Lim Xue; Zafar, Ayesha; Blanco-Cabra, Núria; Torrents, Eduard; Dömötör, Orsolya; May, Nóra V.; Darvasiova, Denisa;
Enyedy, Éva A.; Popović-Bijelić, Ana  ; Reynisson, Jóhannes; Rapta, Peter; Babak, Maria V.; Pastorin, Giorgia; Arion, Vladimir B.;

Bicyclic α-Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer's Disease   [2020]

Abás, Sònia; Rodríguez-Arévalo, Sergio; Bagán, Andrea; Griñán-Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins, Elies; Luque, F. Javier;
Pérez-Lozano, Pilar; De Jonghe, Steven; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, M. Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica  ; Đikić, Teodora  ; Nikolić, Katarina  ; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmen;

A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype a metalloprotease (✓)   [2007]

Burnett, James C.; Opsenica, Dejan M.  ; Sriraghavan, Kamaraj; Panchal, Rekha G.; Ruthel, Gordon; Hermone, Ann R.; Nguyen, Tam L.; Kenny, Tara A.; Lane, Douglas J.; McGrath, Connor F.;
Schmidt, James J.; Vennerstrom, Jonathan L.; Gussio, Rick; Šolaja, Bogdan A. ; Bavari, Sina;

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