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New Iron Twist to Chloroquine─Upgrading Antimalarials with Immunomodulatory and Antimicrobial Features   [2023]

Jelena Aksić  ; Marija Genčić  ; Nikola Stojanović ; Niko Radulovic  ; Dragan Zlatković  ; Marina Dimitrijević  ; Zorica Stojanović-Radić  ; Jelena Srbljanović  ; Tijana Štajner  ; Ljiljana Jovanović

Bicyclic α-Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer's Disease   [2020]

Abás, Sònia; Rodríguez-Arévalo, Sergio; Bagán, Andrea; Griñán-Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins, Elies; Luque, F. Javier;
Pérez-Lozano, Pilar; De Jonghe, Steven; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, M. Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica  ; Đikić, Teodora ; Nikolić, Katarina  ; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmen;

A Chemotype That Inhibits Three Unrelated Pathogenic Targets: The Botulinum Neurotoxin Serotype A Light Chain, P. falciparum Malaria, and the Ebola Filovirus   [2011]

Opsenica, Igor  ; Burnett, James C.; Gussio, Rick; Opsenica, Dejan M.  ; Todorović, Nina  ; Lanteri, Charlotte A.; Sciotti, Richard J.; Gettayacamin, Montip; Basilico, Nicoletta; Taramelli, Donatella;
Nuss, Jonathan E.; Wanner, Laura; Panchal, Rekha G.; Šolaja, Bogdan A. ; Bavari, Sina;

A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype a metalloprotease   [2007]

Burnett, James C.; Opsenica, Dejan M.  ; Sriraghavan, Kamaraj; Panchal, Rekha G.; Ruthel, Gordon; Hermone, Ann R.; Nguyen, Tam L.; Kenny, Tara A.; Lane, Douglas J.; McGrath, Connor F.;
Schmidt, James J.; Vennerstrom, Jonathan L.; Gussio, Rick; Šolaja, Bogdan A. ; Bavari, Sina;

Beyond H2S and NO Interplay: Hydrogen Sulfide and Nitroprusside React Directly to Give Nitroxyl (HNO). A New Pharmacological Source of HNO   [2013]

Filipović, Milos R; Eberhardt, Mirjam; Prokopović, Vladimir; Mijušković, Ana ; Reeh, Peter; Oreščanin Dušić, Zorana  ; Ivanović-Burmazović, Ivana S

An Improved PDE6D Inhibitor Combines with Sildenafil To Inhibit KRAS Mutant Cancer Cell Growth   [2024]

Kaya, Pelin; Schaffner-Reckinger, Elisabeth; Manoharan, Ganesh babu; Vukić, Vladimir  ; Kiriazis, Alexandros; Ledda, Mirko; Burgos Renedo, Maria; Pavić, Karolina; Gaigneaux, Anthoula; Glaab, Enrico;
Kwaku Abankwa, Daniel;

Antioxidant-inspired drug discovery: antitumor metabolite is formed in situ from a hydroxycinnamic acid derivative upon free radical scavenging.   [2019]

Fási, Laura; Di Meo, Florent; Kuo, Ching-Ying; Stojković Burić, Sonja ; Martins, Ana; Kúsz, Norbert; Béni, Zoltán; Dékány, Miklós; Balogh, György Tibor; Pešić, Milica  ;
Wang, Hui-Chun; Trouillas, Patrick; Hunyadi, Attila;

Second Generation Steroidal 4-Aminoquinolines Are Potent, Dual-Target Inhibitors of the Botulinum Neurotoxin Serotype A Metalloprotease and P. falciparum Malaria   [2014]

Videnović, Milica  ; Opsenica, Dejan M.  ; Burnett, James C.; Gomba, Laura; Nuss, Jonathan E.; Selaković, Života  ; Konstantinović, Jelena M.  ; Krstić-Ristivojević, Maja  ; Šegan, Sandra B.  ; Zlatović, Mario  ;
Sciotti, Richard J.; Bavari, Sina; Šolaja, Bogdan A. ;

Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model   [2020]

Horatscheck, Andre; Andrijevic, Ana  ; Nchinda, Aloysius T.; Le Manach, Claire; Paquet, Tanya; Khonde, Lutete Peguy; Dam, Jean; Pawar, Kailash; Taylor, Dale; Lawrence, Nina;
Brunschwig, Christel; Gibhard, Liezl; Njoroge, Mathew; Reader, Janette; van der Watt, Mariette; Wicht, Kathryn; de Sousa, Ana Carolina C.; Okombo, John; Maepa, Keletso; Egan, Timothy J.; Birkholtz, Lyn-Marie; Basarab, Gregory S.; Wittlin, Sergio; Fish, Paul, V; Street, Leslie J.; Duffy, James; Chibale, Kelly;

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