eNauka - pregled

Pregled prema Projekat Bihejvioralni efekti ponavljane primene novosintetisanih supstanci selektivnih za pojedine podtipove benzodiazepinskog mesta vezivanja GABA A receptora: poređenje sa standardnim psihofarmakološkim lekovima (RS-175076)

Prikaz rezultata 1 do 20 od 28  sledeće >
GodinaNaslovAutor(i)Tip rezultataMp-kat.
2018Attaining in vivo selectivity of positive modulation of alpha 3 ss gamma 2 GABA(A) receptors in rats: A hard task!Batinić, Bojan ; Stanković, Tamara; Stephen, Michael; Kodali, Revathi; Tiruveedhula, Veera V.; Li, Guanguan; Scholze, Petra; Marković, Bojan  ; Obradović, Aleksandar; Ernst, Margot;
Cook, James M.; Savić, Miroslav  ;
Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2017Atypical sympathomimetic drug lerimazoline mediates contractile effects in rat aorta predominantly by 5-HT2A receptorsRizvic, Eldina; Jankovic, Goran  ; Kostić Rajačić, Slađana  ; Savić, Miroslav M.  Naučni članak
23M23 - Rad u međ. časopisu
2013Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α 1 GABA A receptorsJoksimović, Srđan; Divljaković, Jovana; van Linn, Michael; Varagić, Zdravko; Brajković, Gordana; Milinković, Marija M.  ; Yin, Wenyuan; Timić, Tamara ; Sieghart, Werner; Cook, James M.;
Savić, Miroslav  ;
Naučni članak
21aM21a - Rad u međ. časopisu izuzetnih vrednosti
2015Biocompatible microemulsions of a model NSAID for skin delivery: A decisive role of surfactants in skin penetration/irritation profiles and pharmacokinetic performance (✓)Todosijević, Marija; Savić, Miroslav M.  ; Batinić, Bojan B. ; Marković, Bojan D.  ; Gasperlin, Mirjana; Randjelović, Danijela  ; Lukić, Milica  ; Savić, Snežana D.  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2014Duration of treatment and activation of alpha(1)-containing GABA(A) receptors variably affect the level of anxiety and seizure susceptibility after diazepam withdrawal in ratsKovacević, Jovana; Timić, Tamara ; Tiruveedhula, Veera V.; Batinić, Bojan ; Namjoshi, Ojas A.; Milić, Marija  ; Joksimović, Srđan; Cook, James M.; Savić, Miroslav  Naučni članak
22M22 - Rad u istaknutom međ. časopisu
2017Elucidation of the profound antagonism of contractile action of phenylephrine in rat aorta effected by an atypical sympathomimetic decongestantRizvić, Eldina; Janković, Goran  ; Savić, Miroslav  Naučni članak
22M22 - Rad u istaknutom međ. časopisu
2016Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABA(A) receptors containing the alpha 5 subunitTimić-Stamenić, Tamara ; Poe, Michael M.; Rehman, Sabah; Santrač, Anja; Divović, Branka  ; Scholze, Petra; Ernst, Margot; Cook, James M.; Savić, Miroslav  Naučni članak
22M22 - Rad u istaknutom međ. časopisu
2013Experimental Design in Formulation of Diazepam Nanoemulsions: Physicochemical and Pharmacokinetic Performances (✓)Đorđević, Sanela M.  ; Radulović, Tamara S.; Cekić, Nebojša  ; Randjelović, Danijela  ; Savić, Miroslav M.  ; Krajišnik, Danina R.  ; Milić, Jela R.  ; Savić, Snežana D.  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2018International Union of Basic and Clinical Pharmacology. CVI: GABAA Receptor Subtype- and Function-selective Ligands: Key Issues in Translation to HumansSieghart, Werner; Savić, Miroslav  Naučni članak
21aM21a - Rad u međ. časopisu izuzetnih vrednosti
2016Lipopolysaccharide exposure during late embryogenesis results in diminished locomotor activity and amphetamine response in females and spatial cognition impairment in males in adult, but not adolescent rat offspringBatinić, Bojan ; Santrač, Anja; Divović, Branka  ; Timić, Tamara ; Stanković, Tamara ; Obradović, Aleksandar; Joksimović, Srđan; Savić, Miroslav  Naučni članak
22M22 - Rad u istaknutom međ. časopisu
2022Metabolism, pharmacokinetics, and anticonvulsant activity of a deuterated analog of the α2/3-selective GABAkine KRM-II-81Golani, Lalit; Divović, Branka  ; Sharmin, Dishary; Pandey, Kamal; Mian, Md Yeunus; Cerne, Rok; Zahn, Nicolas; Meyer, Michelle; Tiruveedhula, Veera; Smith, Jodi;
Ping, Xingjie; Jin, Xiaoming; Lippa, Arnold; Schkeryantz, Jeffrey; Arnold, Leggy; Cook, James; Savić, Miroslav  ; Witkin, Jeffrey;
Naučni članak
23M23 - Rad u međ. časopisu
2013Midazolam impairs acquisition and retrieval, but not consolidation of reference memory in the Morris water mazeTimić, Tamara ; Joksimović, Srđan; Milić, Marija; Divljaković, Jovana; Batinić, Bojan ; Savić, Miroslav  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2020Nanocrystal dispersion of DK-I-56–1, a poorly soluble pyrazoloquinolinone positive modulator of α6 GABAA receptors: Formulation approach toward improved in vivo performance (✓)Mitrović, Jelena ; Divović, Branka  ; Knutson, Daniel; Đoković, Jelena  ; Vulić, Predrag; Randjelović, Danijela  ; Dobričić, Vladimir  ; Čalija, Bojan ; Cook, James; Savić, Miroslav M.  ;
Savić, Snežana  ;
Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2015Negative modulation of alpha(5) GABA(A) receptors in rats may partially prevent memory impairment induced by MK-801, but not amphetamine- or MK-801-elicited hyperlocomotionTimić-Stamenić, Tamara ; Joksimović, Srđan; Biawat, Poonam; Stanković, Tamara ; Marković, Bojan  ; Cook, James M.; Savić, Miroslav  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2015Parenteral nanoemulsions as promising carriers for brain delivery of risperidone: Design, characterization and in vivo pharmacokinetic evaluation (✓)Djordjevic, Sanela M  ; Cekic, Nebojsa  ; Savić, Miroslav M.  ; Isailovic, Tanja M  ; Randjelović, Danijela  ; Marković, Bojan D.  ; Savić, Saša R.  ; Stamenic, Tamara Timic ; Daniels, Rolf; Savić, Snežana D.  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2017Positive modulation of alpha 5 GABA(A) receptors in preadolescence prevents reduced locomotor response to amphetamine in adult female but not male rats prenatally exposed to lipopolysaccharideBatinić, Bojan ; Santrač, Anja; Jančić, Ivan  ; Li, Guanguan; Vidojević, Aleksandra  ; Marković, Bojan  ; Cook, James M.; Savić, Miroslav  Naučni članak
22M22 - Rad u istaknutom međ. časopisu
2022Postweaning positive modulation of α5GABAA receptors improves autism-like features in prenatal valproate rat model in a sex-specific manner (✓)Santrač, Anja; Bijelić, Dunja  ; Stevanović, Vladimir; Banićević, Marija; Aranđelović, Jovana  ; Batinić, Bojan ; Sharmin, Dishary; Cook, James; Savić, Miroslav  Naučni članak
21aM21a - Rad u međ. časopisu izuzetnih vrednosti
2013PWZ-029, an inverse agonist selective for alpha(5) GABA(A) receptors, improves object recognition, but not water-maze memory in normal and scopolamine-treated ratsMilić, Marija; Timić, Tamara ; Joksimović, Srđan; Biawat, Poonam; Rallapalli, Sundari; Divljaković, Jovana; Radulović, Tamara; Cook, James M.; Savić, Miroslav  Naučni članak
21M21 - Rad u vrhunskom međ. časopisu
2019Selektivna modulacija GABAA receptora koji sadrže alfa6 podjedinicu na eksperimentalnom modelu trigeminalnog neuropatskog bolaVasović, Dina  Doktorska disertacija
70M70 - Odbranjena doktorska disertacija
2015Uticaj modulacije GABAA receptora koji sadrže [alfa] 5 podjedinicu na poremećaje ponašanja pacova izazvane primenom dizocilpina, skopolamina i amfetaminaTimić Stamenić, Tamara S.Doktorska disertacija
70M70 - Odbranjena doktorska disertacija