| Title: | Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy |
Authors: | Jovanović, Mirna ; Zhukovsky, Daniil; Podolski-Renić, Ana ; Domračeva, Ilona; Žalubovskis, Raivis; Senćanski, Milan V. ; Glišić, Sanja ; Sharoyko, Vladimir; Tennikova, Tatiana; Dar'in, Dmitry;
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Issue Date: | 2019 |
Publication: | European Journal of Medicinal Chemistry |
ISSN: | 0223-5234 European Journal of Medicinal Chemistry Search Idenfier |
Type: | Article |
Collation: | vol. 181 str. 111580-111580 |
DOI: | 10.1016/j.ejmech.2019.111580 |
WoS-ID: | 000493211900034 |
Scopus-ID: | 2-s2.0-85073183701 |
PMID: | 31400708 |
URI: | https://vinar.vin.bg.ac.rs/handle/123456789/8532 https://www.sciencedirect.com/science/article/pii/S0223523419307147?via%3Dihub https://enauka.gov.rs/handle/123456789/503502 https://radar.ibiss.bg.ac.rs/handle/123456789/3488 |
Project: | Russian Foundation for Basic Research (RFBR) [18-515-76001] Identifikacija molekularnih markera za predikciju progresije tumora, odgovora na terapiju i ishoda bolesti (RS-41031) ERA.Net RUS plus joint program grant [RUS_ST2017-309] State Education Development Agency of Republic of Latvia ["THIOREDIN"] Short-Term Scientific Mission (STSM) Grant from COST Action "New diagnostic and therapeutic tools against multidrug resistant tumors" [CA17104] European Cooperation in Science and Technology (COST) |
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