| Назив: | From PROTAC to inhibitor: Structure-guided discovery of potent and orally bioavailable BET inhibitors |
Аутори: | Koravović, Mladen   ; Mayasundari, Anand; Tasić, Gordana ; Keramatnia, F.; Stachowski, Timothy R.; Cui, Huarui; Chai, Sergio C.; Jonchere, Barbara; Yang, Lei; Li, Yong;
Fu, Xiang; Hiltenbrand, Ryan; Paul, Leena; Mishra, Vibhor; Klco, Jeffery M.; Roussel, Martine F.; Pomerantz, William CK.; Fischer, Marcus; Ranković, Zoran; Savić, Vladimir ;
|
Година: | 2023 |
Публикација: | European Journal of Medicinal Chemistry |
ISSN: | 0223-5234 European Journal of Medicinal Chemistry Претражи идентификатор |
Издавач: | Elsevier Masson s.r.l. |
Тип резултата: | Научни чланак |
Колација: | vol. 251 str. 115246-115246 |
DOI: | 10.1016/j.ejmech.2023.115246 |
WoS-ID: | 000952151800001 |
Scopus-ID: | 2-s2.0-85149446323 |
PMID: | 36898329 |
PMCID: | PMC10165889 |
URI: | https://farfar.pharmacy.bg.ac.rs/handle/123456789/4513
https://enauka.gov.rs/handle/123456789/605289 |
Пројекат: | ALSAC and R35GM142772 (to MF)
R35GM140837 (to WCKP)
Crystallographic data were collected at
Southeast Regional Collaborative Access Team (SER-CAT) 22-ID beam-
line at the Advanced Photon Source, Argonne National Laboratory.
SER-CAT is supported by its member institutions, and equipment grants
(S10_RR25528, S10_RR028976 and S10_OD027000) from the National
Institutes of Health.
The Advanced Photon Source was supported
by the U. S. Department of Energy, Office of Science, Office of Basic
Energy Sciences, under Contract No. W-31-109-Eng-38
The Science fund of the Republic of Serbia: program, Diaspora
Grant no: 6463913
Ministarstvo prosvete, nauke i tehnološkog razvoja Republike Srbije, Ugovor br. 200161 (Univerzitet u Beogradu, Farmaceutski fakultet) |
М-категорија: | 21aM21a - Рад у међ. часопису изузетних вредности |
